SCHEMBL19648317

SCHEMBL19648317

O=C(NF)c1c(F)cccc1Cl

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 10/20 0.65
JAK2 O60674 1/20 0.59
JAK1 P23458 1/20 0.59
TYK2 P29597 1/20 0.59
HPGD P15428 1/20 0.57
MAPT P10636 2/20 0.55
LMNA P02545 1/20 0.55
PKM P14618 1/20 0.55
KMT2A Q03164 1/20 0.55
TLR7 Q9NYK1 1/20 0.55
RAB9A P51151 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
POLB P06746 1/20 0.54
ITGB2 P05107 1/20 0.52
ICAM1 P05362 1/20 0.52
ITGAL P20701 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19648319 0.88 ALDH1A1 (0.54) GAAJAK2JAK1TYK2HPGD
SCHEMBL28869679 0.85 GAA (0.65) GAAJAK2JAK1TYK2HPGD
SCHEMBL25051950 0.83 GAA (0.63) GAAJAK2JAK1TYK2HPGD
SCHEMBL14968580 0.83 GAA (0.63) GAAJAK2JAK1TYK2HPGD
SCHEMBL18306503 0.83 GAA (0.63) GAAJAK2JAK1TYK2HPGD
SCHEMBL11100266 0.81 GAA (0.61) GAAJAK2JAK1TYK2MAPT
SCHEMBL11098006 0.81 GAA (0.61) GAAJAK2JAK1TYK2HPGD
Hydrochloric Acid SCHEMBL11098010 0.80 GAA (0.59) GAAJAK2JAK1TYK2MAPT
SCHEMBL11499405 0.80 GAA (0.59) GAAJAK2JAK1TYK2HPGD
SCHEMBL2876974 0.79 GAA (0.58) GAAJAK2JAK1TYK2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2846804-B1 TETRAHYDRONAPHTHYRIDINE AND RELATED BICYCLIC COMPOUNDS FOR INHIBITION OF RORgamma ACTIVITY AND THE TREATMENT OF DISEASE MERCK SHARP & DOHME (US) 2017-11-29 EP disclosed