SCHEMBL1965728

SCHEMBL1965728

COc1cccc(CCN(C)C2CC2)c1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.63
SIGMAR1 Q99720 2/20 0.54
TAAR1 Q96RJ0 1/20 0.53
CHRM2 P08172 2/20 0.50
CHRM1 P11229 2/20 0.50
CHRM3 P20309 2/20 0.50
HRH3 Q9Y5N1 3/20 0.49
ALDH1A1 P00352 1/20 0.48
CALM1 P0DP23 1/20 0.46
CAMKK2 Q96RR4 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1971180 0.84 CALM1 (0.47) AOC3ALDH1A1CALM1KMT2A
SCHEMBL1966332 0.81 AOC3 (0.59) AOC3SIGMAR1TAAR1HRH3
SCHEMBL18122711 0.80 AOC3 (0.75) AOC3SIGMAR1TAAR1CHRM2CHRM1
SCHEMBL44276 0.80 AOC3 (0.75) AOC3SIGMAR1TAAR1CHRM2CHRM1
SCHEMBL1970244 0.80 TAAR1 (0.49) TAAR1HRH3
SCHEMBL18744298 0.79 CALM1 (0.47) AOC3SIGMAR1TAAR1HRH3ALDH1A1
SCHEMBL17470863 0.79 CALM1 (0.47) AOC3SIGMAR1TAAR1HRH3ALDH1A1
SCHEMBL17470861 0.79 CALM1 (0.47) AOC3SIGMAR1TAAR1HRH3ALDH1A1
SCHEMBL17297951 0.79 CALM1 (0.47) AOC3SIGMAR1TAAR1HRH3ALDH1A1
Hydrochloric Acid SCHEMBL8508344 0.79 AOC3 (0.73) AOC3SIGMAR1TAAR1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD. (CH) 2011-09-01 US disclosed
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES HCRTR2, HCRTR1, HRH3 AOC3 550/4885SIGMAR1 108/4885TAAR1 48/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.