SCHEMBL1965745

SCHEMBL1965745

COc1ccccc1CCN(C)C1CC1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.61
SIGMAR1 Q99720 2/20 0.52
HTR2A P28223 1/20 0.51
TAAR1 Q96RJ0 1/20 0.50
ALDH1A1 P00352 2/20 0.48
KCNH2 Q12809 1/20 0.47
HRH3 Q9Y5N1 3/20 0.47
CHRM2 P08172 1/20 0.46
BCHE P06276 1/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
ALOX12 P18054 1/20 0.45
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27366104 0.84 HTR2A (0.67) AOC3SIGMAR1HTR2AALDH1A1CHRM2
SCHEMBL31331990 0.84 HTR2A (0.67) AOC3SIGMAR1HTR2AALDH1A1CHRM2
SCHEMBL1968729 0.80 AOC3 (0.64) AOC3HTR2ATAAR1ALDH1A1
SCHEMBL2937482 0.79 AOC3 (0.73) AOC3SIGMAR1HTR2ATAAR1KCNH2
SCHEMBL1968535 0.78 HTR2A (0.55) HTR2ATAAR1KCNH2
Hydrochloric Acid SCHEMBL8509376 0.78 AOC3 (0.71) AOC3SIGMAR1HTR2ATAAR1ALDH1A1
SCHEMBL27817763 0.77 TAAR1 (0.62) AOC3HTR2ATAAR1KCNH2MEN1
SCHEMBL2404071 0.77 TAAR1 (0.62) AOC3HTR2ATAAR1ALDH1A1CHRM2
SCHEMBL1969126 0.77 HTR6 (0.72) HTR2ABCHE
SCHEMBL31396927 0.77 HTR6 (0.72) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD. (CH) 2011-09-01 US disclosed
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES HCRTR2, HCRTR1, HRH3 AOC3 550/4885SIGMAR1 108/4885HTR2A 46/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.