SCHEMBL1965760

SCHEMBL1965760

O=C(Cc1ccc(Cl)cc1)NC(=O)c1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 16/20 0.55
GSPT1 P15170 4/20 0.48
DDB1 Q16531 2/20 0.48
CYP2C19 P33261 1/20 0.48
KCNH2 Q12809 1/20 0.48
CSNK1A1 P48729 3/20 0.43
IKZF3 Q9UKT9 4/20 0.42
MAPT P10636 2/20 0.42
IKZF1 Q13422 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1963376 0.91 CRBN (0.53) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1962950 0.91 CRBN (0.55) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1962928 0.91 CRBN (0.52) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1961959 0.90 CRBN (0.55) CRBNGSPT1DDB1CSNK1A1IKZF3
SCHEMBL1964617 0.89 CRBN (0.52) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1962557 0.88 CRBN (0.57) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1961984 0.87 CRBN (0.59) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1962957 0.87 CRBN (0.50) CRBNGSPT1DDB1CYP2C19KCNH2
SCHEMBL1962874 0.86 CRBN (0.53) CRBNGSPT1DDB1CSNK1A1IKZF3
SCHEMBL1962830 0.86 CRBN (0.53) CRBNGSPT1DDB1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US claimed
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARM LLC (US) 2020-04-16 US disclosed
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARMACEUTICALS, LLC (US) 2014-10-23 US disclosed
EP-1919892-B1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2013-08-14 EP disclosed
US-8481568-B2 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION (US) 2013-07-09 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885GSPT1 861/4885DDB1 820/4885
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885GSPT1 861/4885DDB1 820/4885
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SI, CYP3A5, CYP2D6 CRBN 2589/4885GSPT1 1740/4885DDB1 4509/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 CRBN 2589/4885GSPT1 1740/4885DDB1 4509/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.