SCHEMBL19658993

SCHEMBL19658993

OC(O)c1nnc2ccc(C(F)(F)F)cn12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 2/20 0.49
HSD17B10 Q99714 1/20 0.49
SCN5A Q14524 8/20 0.46
USP7 Q93009 1/20 0.40
RBP4 P02753 2/20 0.39
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
GFER P55789 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
RCE1 Q9Y256 1/20 0.37
MAPK14 Q16539 3/20 0.35
PIM1 P11309 1/20 0.34
RIPK1 Q13546 1/20 0.34
SCN1A P35498 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11914744 0.83 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL19292586 0.78 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL1189278 0.74 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL11918906 0.74 KDM4E (0.56) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL19659055 0.73 SMN1; SMN2 (0.32) SMN1; SMN2RAB9A
Bromide SCHEMBL1189112 0.72 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL18365954 0.72 RBP4 (0.51) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL19292958 0.71 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL13687300 0.71 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A
SCHEMBL24654157 0.71 SCN5A (0.41) ALDH1A1SMN1; SMN2KDM4EHSD17B10SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017004500-A9 BICYCLIC LACTAMS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2017-11-30 WO disclosed