SCHEMBL19662408

SCHEMBL19662408

Clc1nc(OC2CCCCC2)c2occc2n1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 5/20 0.36
HRH4 Q9H3N8 1/20 0.35
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
JAK3 P52333 2/20 0.33
PTGES O14684 1/20 0.32
LOX P28300 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31
KMO O15229 1/20 0.31
MCHR1 Q99705 2/20 0.31
KDM4C Q9H3R0 1/20 0.30
CNR1 P21554 1/20 0.30
HDAC3 O15379 1/20 0.30
CDK9 P50750 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
PDGFRB P09619 1/20 0.30
PDGFRA P16234 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3704178 0.96 LRRK2 (0.35) LRRK2HRH4PDE4APDE4BPDE4C
SCHEMBL19662401 0.85
SCHEMBL19662404 0.79 IRAK4 (0.46) LRRK2
SCHEMBL29487321 0.76 HRH4 (0.44) HRH4PTGESPDGFRB
SCHEMBL20273951 0.74 KMT2A (0.47) PDE4A
SCHEMBL7601802 0.73 ALDH1A1 (0.37) PDE4APDGFRB
SCHEMBL19663154 0.70 HRH4 (0.40) LRRK2HRH4PDE4APDE4BPDE4C
SCHEMBL19662572 0.70 IRAK4 (0.60)
SCHEMBL3712626 0.70 IRAK4 (0.44) LRRK2PDE4A
SCHEMBL1709800 0.69 IRAK4 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017205766-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed