SCHEMBL19663154

SCHEMBL19663154

Clc1nc(OC2CCCCC2)c2ncccc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
LRRK2 Q5S007 4/20 0.39
PDE5A O76074 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
PTGES O14684 1/20 0.35
SLC40A1 Q9NP59 1/20 0.35
MCHR1 Q99705 2/20 0.35
JAK3 P52333 2/20 0.35
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
GRM5 P41594 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19644121 0.79 ROCK2 (0.35)
SCHEMBL19662554 0.79 IRAK4 (0.47) HRH3
SCHEMBL29487321 0.78 HRH4 (0.44) HRH4PDE5AHRH3PTGESKDM4E
SCHEMBL23107674 0.72 LRRK2 (0.41) HRH4LRRK2FFAR4PTGESSLC40A1
SCHEMBL22872852 0.72 KMT2A (0.49) PDE5AKDM4ECDK7CDK9
SCHEMBL19662557 0.71 IRAK4 (0.56)
SCHEMBL38659897 0.71 PRMT5 (0.37) HRH4KDM4EL3MBTL1
SCHEMBL22411411 0.70 KMT2A (0.47) PDE5AKDM4ECDK7CDK9
SCHEMBL3024650 0.70 JAK3 (0.42) LRRK2PTGESJAK3CDK9
SCHEMBL30872619 0.70 JAK3 (0.42) LRRK2PTGESJAK3CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017205766-A1 INHIBITORS OF INTERLEUKIN-1 RECEPTOR-ASSOCIATED KINASE PHARMACYCLICS LLC (US) 2017-11-30 WO disclosed