SCHEMBL19665014

SCHEMBL19665014

Cc1cccc2cc(-c3cc(C(F)(F)F)nn3-c3ccc(NS(N)(=O)=O)cc3)ccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 7/20 0.61
PTGS2 P35354 13/20 0.56
PTGS1 P23219 6/20 0.55
PTGES O14684 1/20 0.53
HDAC3 O15379 1/20 0.53
CA12 O43570 1/20 0.53
PDE5A O76074 1/20 0.53
ABCB11 O95342 1/20 0.53
MT-CO2 P00403 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
LMNA P02545 1/20 0.53
CA3 P07451 1/20 0.53
CYP3A4 P08684 1/20 0.53
ALOX5 P09917 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
ADRB3 P13945 1/20 0.53
ALOX15 P16050 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718293 0.89 PDPK1 (0.78) PDPK1PTGS2CA9
SCHEMBL15346826 0.86 PDPK1 (0.77) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL2732571 0.85 PDPK1 (0.72) PDPK1PTGS2PTGS1CYP2C9
SCHEMBL15347056 0.85 PTGS2 (0.63) PDPK1PTGS2PTGS1PTGESHDAC3
SCHEMBL15347135 0.85 PTGS2 (0.64) PDPK1PTGS2PTGS1PTGESHDAC3
SCHEMBL15346636 0.83 PDPK1 (0.70) PDPK1PTGS2PTGS1
SCHEMBL2720059 0.83 PTGS2 (0.75) PDPK1PTGS2PTGS1PTGESHDAC3
SCHEMBL15346929 0.82 PDPK1 (0.76) PDPK1PTGS2PTGS1PTGESHDAC3
SCHEMBL15347122 0.82 PDPK1 (0.78) PDPK1PTGS2PTGS1HDAC3HDAC4
SCHEMBL15346937 0.81 PDPK1 (0.62) PDPK1PTGS2PTGS1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635274-B1 ANTI-STAPHYLOCOCCAL CELECOXIB DERIVATIVES UNIV OHIO STATE RES FOUND (US) 2017-12-06 EP disclosed