SCHEMBL19669752

SCHEMBL19669752

C=C(Cl)C(=O)NC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
EPHX1 P07099 1/20 0.34
KDM4E B2RXH2 4/20 0.34
RAB9A P51151 2/20 0.34
CYP2C9 P11712 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
EPHX2 P34913 1/20 0.32
IMPDH2 P12268 1/20 0.31
IMPDH1 P20839 1/20 0.31
APEX1 P27695 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22366261 0.80 LMNA (0.39) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL6859267 0.76 KDM4E (0.46) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL13588042 0.76 EPHX1 (0.36) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL9171219 0.76 ALDH1A1 (0.36) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL138082 0.76 EPHX1 (0.41) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL29088791 0.74 TDP1 (0.35) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL9242168 0.74 EPHX1 (0.39) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL19669753 0.74 EPHX1 (0.34) LMNAEPHX1KDM4ERAB9ACYP2C9
Dimethylamine SCHEMBL27557791 0.72 EPHX1 (0.38) LMNAEPHX1KDM4ERAB9ACYP2C9
SCHEMBL5219501 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834571-B2 Compounds for inhibiting cell proliferation in EGFR-driven cancers ARIAD PHARMACEUTICALS, INC. (US) 2017-12-05 US disclosed