SCHEMBL19672008

SCHEMBL19672008

CC(=N)c1cc(Br)c(F)cc1NC(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNK2 O95069 1/20 0.34
KCNK10 P57789 1/20 0.34
VNN1 O95497 1/20 0.32
KCNN4 O15554 2/20 0.32
HDAC6 Q9UBN7 1/20 0.30
TAS2R14 Q9NYV8 1/20 0.30
GPR27 Q9NS67 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19671926 0.78 VNN1 (0.32) KCNK2KCNK10VNN1HDAC6
SCHEMBL19672102 0.76 VNN1 (0.31) KCNK2KCNK10VNN1
SCHEMBL21416790 0.76 KCNN4 (0.32) VNN1KCNN4HDAC6
SCHEMBL20418717 0.73 VNN1 (0.32) VNN1KCNN4
SCHEMBL19671910 0.71 LRRK2 (0.31)
SCHEMBL19672014 0.70 PIK3CA (0.43)
SCHEMBL3182764 0.69 KDM1A (0.32)
SCHEMBL19671830 0.68 ALDH1A1 (0.46)
SCHEMBL19416920 0.68
SCHEMBL19671998 0.67 KAT6A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964221-B1 COMPOUNDS INHIBITING LEUCINE-RICH REPEAT KINASE ENZYME ACTIVITY MERCK SHARP & DOHME (US) 2017-12-06 EP disclosed