SCHEMBL196747

SCHEMBL196747

O=C(Nc1cc(Nc2ccc(Cl)c(Cl)c2)nc2ccccc12)c1ccco1.O=C(Nc1cc(Nc2ccccc2)nc2ccccc12)C1CCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 10/20 0.48
NPC1 O15118 8/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
MAPT P10636 8/20 0.47
KDM4E B2RXH2 5/20 0.47
ALDH1A1 P00352 5/20 0.47
USP2 O75604 1/20 0.47
MAPK8 P45983 1/20 0.46
MAPK10 P53779 1/20 0.46
TP53 P04637 3/20 0.46
LMNA P02545 4/20 0.44
POLB P06746 3/20 0.44
TSHR P16473 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL196069 0.90 RAB9A (0.59) RAB9ANPC1CASP3SENP8SENP7
SCHEMBL196452 0.88 GRM4 (0.47) RAB9ANPC1MAPTALDH1A1TP53
SCHEMBL196377 0.86 GRM4 (0.49) RAB9ANPC1MAPTTP53RXFP1
SCHEMBL196780 0.85 GRM4 (0.51) RAB9ANPC1MAPTTP53RXFP1
SCHEMBL29501836 0.85 GRM4 (0.51) RAB9ANPC1MAPTTP53RXFP1
SCHEMBL30637139 0.85 GRM4 (0.51) RAB9ANPC1MAPTTP53RXFP1
SCHEMBL197210 0.83 MAPK8 (0.58) RAB9ANPC1MAPTKDM4EALDH1A1
SCHEMBL196310 0.82 RXFP1 (0.47) RAB9ANPC1MAPTTP53KMT2A
SCHEMBL196512 0.81 MAPT (0.55) RAB9ANPC1MAPTALDH1A1MAPK8
SCHEMBL197113 0.80 MAPT (0.57) RAB9AMAPTKDM4EALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2012500255-A 2012-01-05 JP claimed
EP-2323661-A1 A3 ADENOSINE RECEPTOR ALLOSTERIC MODULATORS Universiteit Leiden (NL) 2011-05-25 EP claimed
EP-2323661-A1 A3 ADENOSINE RECEPTOR ALLOSTERIC MODULATORS Universiteit Leiden (NL) 2011-05-25 EP disclosed