SCHEMBL19675175

SCHEMBL19675175

COCc1cccc(N(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
MAOB P27338 1/20 0.40
FFAR1 O14842 1/20 0.38
AGXT P21549 3/20 0.38
SIGMAR1 Q99720 2/20 0.38
GRM2 Q14416 1/20 0.38
BCHE P06276 1/20 0.37
IDO1 P14902 2/20 0.37
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.37
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13681219 1.00 TSHR (0.40) TSHRMAOBFFAR1AGXTSIGMAR1
SCHEMBL28874019 0.88 TSHR (0.46) TSHRMAOBAGXTBCHEIDO1
SCHEMBL279614 0.82 ALDH1A1 (0.45) TSHRAGXTBCHEIDO1TP53
SCHEMBL279615 0.82 ALDH1A1 (0.45) TSHRAGXTBCHEIDO1TP53
SCHEMBL791873 0.81 ALDH1A1 (0.50) TSHRAGXTIDO1KDM4EALDH1A1
SCHEMBL12957222 0.80 TP53 (0.54) TSHRSIGMAR1TP53CYP1A2CYP2D6
SCHEMBL13136839 0.79 TP53 (0.52) TSHRSIGMAR1TP53KDM4EALDH1A1
SCHEMBL76603 0.79 TP53 (0.52) TSHRSIGMAR1TP53KDM4EALDH1A1
SCHEMBL10330363 0.78 IDO1 (0.46) AGXTIDO1KDM4EALDH1A1CYP1A2
SCHEMBL487468 0.77 IDO1 (0.48) MAOBFFAR1AGXTIDO1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2448925-B1 EMISSIVE ARYL-HETEROARYL COMPOUNDS NITTO DENKO CORP (JP) 2017-12-06 EP disclosed