SCHEMBL19682377

SCHEMBL19682377

Cc1ccc(F)c([C@H](C)[C@@H](N)C(=O)O)c1C

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 16/20 0.36
CHRM1 P11229 16/20 0.36
RRM1 P23921 16/20 0.36
RRM2B Q7LG56 16/20 0.36
SLC7A5 Q01650 1/20 0.35
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 2/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
SLC1A1 P43005 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19682546 1.00 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL30298149 1.00 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL19682547 1.00 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL19682740 1.00 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL19682386 1.00 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
Hydrochloric Acid SCHEMBL30821884 0.98 CHRM2 (0.36) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL20889297 0.90 SLC7A5 (0.38) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL19682581 0.90 SLC7A5 (0.38) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL20872565 0.87 NR1I2 (0.38) CHRM2CHRM1RRM1RRM2BSLC7A5
SCHEMBL19682387 0.87 NR1I2 (0.38) CHRM2CHRM1RRM1RRM2BSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 CHRM2 4302/4885CHRM1 4399/4885RRM1 5/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B CHRM2 4208/4885CHRM1 4101/4885RRM1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.