SCHEMBL19682687

SCHEMBL19682687

CSc1nc(=O)c2c(ncn2CC(C)(C)O)n1Cc1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
BRD4 O60885 3/20 0.44
BRD2 P25440 1/20 0.44
BRD3 Q15059 1/20 0.44
BRDT Q58F21 1/20 0.44
MAPK1 P28482 3/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 4/20 0.40
TSHR P16473 5/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 3/20 0.37
HPGD P15428 2/20 0.37
TP53 P04637 1/20 0.37
XBP1 P17861 1/20 0.37
P2RX3 P56373 3/20 0.36
BRAF P15056 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814682 0.86 BRD4 (0.60) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL19682689 0.82 ATM (0.46) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL17814708 0.82 KMT2A (0.47) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL19682686 0.79 P2RX3 (0.45) P2RX3
SCHEMBL17814707 0.77 ATM (0.49) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL19682688 0.72 P2RX3 (0.60) P2RX3
SCHEMBL19682474 0.72 P2RX3 (0.56) P2RX3
SCHEMBL19683047 0.70 P2RX3 (0.61) P2RX3
SCHEMBL19682695 0.70 P2RX3 (0.56) P2RX3
SCHEMBL30804835 0.70 ATM (0.52) ATMAPOBEC3GBRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed