SCHEMBL19682689

SCHEMBL19682689

CSc1nc(=O)c2c(ncn2CC(F)F)n1Cc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
BRD4 O60885 2/20 0.45
BRD2 P25440 1/20 0.45
BRD3 Q15059 1/20 0.45
BRDT Q58F21 1/20 0.45
MAPK1 P28482 3/20 0.41
LMNA P02545 2/20 0.41
KMT2A Q03164 4/20 0.40
TSHR P16473 5/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
P2RX3 P56373 1/20 0.38
MEN1 O00255 3/20 0.38
HPGD P15428 2/20 0.38
GAA P10253 1/20 0.38
PKM P14618 1/20 0.38
TP53 P04637 3/20 0.36
XBP1 P17861 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17814682 0.87 BRD4 (0.60) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL19682687 0.82 ATM (0.45) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL17814708 0.81 KMT2A (0.47) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL17814707 0.77 ATM (0.49) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL30804853 0.72 P2RX3 (0.40) BRD4BRD2BRD3BRDTP2RX3
SCHEMBL28543995 0.72 P2RX3 (0.40) BRD4BRD2BRD3BRDTP2RX3
SCHEMBL19682690 0.72 P2RX3 (0.60) P2RX3
SCHEMBL19683040 0.72 P2RX3 (0.57) P2RX3
SCHEMBL30804835 0.71 ATM (0.52) ATMAPOBEC3GBRD4BRD2BRD3
SCHEMBL17814709 0.71 PNP (0.54) ATMAPOBEC3GMAPK1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112409331-B Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-02-20 CN disclosed
CN-112409331-A Heterocyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-02-26 CN disclosed
WO-2017209267-A1 PURINE DERIVATIVE 塩野義製薬株式会社 2017-12-07 WO disclosed