SCHEMBL19684294

SCHEMBL19684294

COC(=O)[C@@H](NC(=O)c1ccc(C#CC#Cc2ccccc2N)cc1)C(C)(O)C(F)F

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.33
CTSG P08311 1/20 0.33
CTRB1 P17538 1/20 0.33
CMA1 P23946 1/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15235718 1.00 PRSS1 (0.33) PRSS1CTSGCTRB1CMA1HTT
SCHEMBL254843 0.94 KDM4E (0.37)
SCHEMBL15235717 0.90 PRSS1 (0.35) PRSS1CTSGCTRB1CMA1LMNA
SCHEMBL19684183 0.88
SCHEMBL15227262 0.88
SCHEMBL255321 0.88
SCHEMBL15235715 0.88 PRSS1 (0.35) PRSS1CTSGCTRB1CMA1
SCHEMBL15237903 0.88 LMNA (0.36) LMNAL3MBTL1TSHR
SCHEMBL255216 0.83 KDM4E (0.40)
SCHEMBL19684184 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170349544-A1 Ethynylbenzene Derivatives DUKE UNIVERSITY 2017-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170349544-A1 Ethynylbenzene Derivatives Q6ZSR9, EPX, ZYX PRSS1 1288/4885CTSG 3126/4885CTRB1 580/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.