SCHEMBL19696802

SCHEMBL19696802

N[C@H](C(=O)O)[C@H](c1ccc(F)cc1)c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC1A1 P43005 2/20 0.49
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
EPHX1 P07099 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
SLC6A9 P48067 2/20 0.40
SLC6A5 Q9Y345 2/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19696914 0.94 SLC1A1 (0.54) SLC1A1HDAC4HDAC7HDAC5CES2
SCHEMBL22088893 0.90 SLC1A1 (0.46) SLC1A1HDAC4HDAC7HDAC5CES2
SCHEMBL19696805 0.90 SLC1A1 (0.46) SLC1A1HDAC4HDAC7HDAC5CES2
SCHEMBL7103759 0.89 LMNA (0.45) SLC1A1EPHX1CNR2
SCHEMBL7103757 0.89 LMNA (0.45) SLC1A1EPHX1CNR2
SCHEMBL4799034 0.87 SLC1A1 (0.47) SLC1A1HDAC4HDAC7HDAC5
SCHEMBL3164836 0.87 SLC1A1 (0.47) SLC1A1HDAC4HDAC7HDAC5
SCHEMBL18627316 0.85 SLC1A1 (0.42) SLC1A1HDAC4HDAC7HDAC5CES2
Hydrochloric Acid SCHEMBL4798059 0.85 SLC1A1 (0.46) SLC1A1HDAC4HDAC7HDAC5IDO1
SCHEMBL18627259 0.84 SLC1A3 (0.46) SLC1A1CES2EPHX1IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9840478-B2 Piperazine derivatives as HIV protease inhibitors MERCK SHARP & DOHME CORP. (US) 2017-12-12 US disclosed