SCHEMBL1969954

SCHEMBL1969954

NCCC(=O)[C@@H]1CCCN1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
PRCP P42785 2/20 0.39
DPP4 P27487 4/20 0.39
GLI1 P08151 1/20 0.38
DPP8 Q6V1X1 2/20 0.38
DPP9 Q86TI2 2/20 0.38
SCN4A P35499 1/20 0.37
DPP7 Q9UHL4 2/20 0.37
FAP Q12884 1/20 0.37
CTSC P53634 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 1/20 0.34
MEN1 O00255 1/20 0.34
BLM P54132 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL514066 0.83
SCHEMBL514065 0.83
SCHEMBL6894328 0.83 NOS2 (0.37) NOS2NOS3NOS1PRCPDPP4
SCHEMBL7432758 0.82 NOS2 (0.48) NOS2NOS3NOS1PRCPDPP4
SCHEMBL2645121 0.80 PRCP (0.50) NOS2NOS3NOS1PRCPDPP4
SCHEMBL30973638 0.80 PRCP (0.50) NOS2NOS3NOS1PRCPDPP4
SCHEMBL4685705 0.80 NOS2 (0.41) NOS2NOS3NOS1PRCPDPP4
Proline SCHEMBL17294497 0.79 NOS2 (0.41) NOS2NOS3NOS1PRCPDPP4
Propionic Acid SCHEMBL29167414 0.79 PRCP (0.36) NOS2NOS3NOS1PRCPHDAC3
SCHEMBL8062198 0.79 NOS2 (0.46) NOS2NOS3NOS1PRCPDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450841-A4 TRI-, TETRA-, AND PENTA-PEPTIDES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LAB (US) 2007-01-24 EP claimed
US-7037897-B2 TRI-, TETRA-, and penta-peptides having antiangiogenic activity ABBOTT LABORATORIES (US) 2006-05-02 US claimed
EP-1450841-A2 TRI-, TETRA-, AND PENTA-PEPTIDES HAVING ANTIANGIOGENIC ACTIVITY Abbott Laboratories (US) 2004-09-01 EP claimed
US-20030109456-A1 TRI-, TETRA-, and penta-peptides having antiangiogenic activity ABBVIE INC. 2003-06-12 US claimed
WO-2003037912-A2 TRI-, TETRA-, AND PENTA-PEPTIDES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LABORATORIES (US) 2003-05-08 WO claimed
US-4318905-A Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues SYNTEX (U.S.A.) INC. (US) 1982-03-09 US claimed
EP-2177530-B1 Octapeptide having antiangiogenic activity ABBOTT LAB (US) 2011-06-22 EP disclosed
EP-2177530-A1 Octapeptide having antiangiogenic activity Abbott Laboratories (US) 2010-04-21 EP disclosed
US-20080071062-A1 TETRA-, PENTA-, HEXA- AND HEPTAPEPTIDES HAVING ANTIANGIOGENIC ACTIVITY HAVIV FORTUNA 2008-03-20 US disclosed
US-20070167376-A1 Hexa-, Hepta-, and Octapeptides Having Antiangiogenic Activity HAVIV FORTUNA 2007-07-19 US disclosed
US-7169888-B2 Tetra-, penta-, hexa- and heptapeptides having antiangiogenic activity ABBOTT LABORATORIES (US) 2007-01-30 US disclosed
EP-1450841-A4 TRI-, TETRA-, AND PENTA-PEPTIDES HAVING ANTIANGIOGENIC ACTIVITY ABBOTT LAB (US) 2007-01-24 EP disclosed
US-7122625-B2 Hexa-, hepta-, and octapeptides having antiangiogenic activity ABBOTT LABORATORIES (US) 2006-10-17 US disclosed
EP-0021234-B1 NONAPEPTIDE AND DECAPEPTIDE DERIVATIVES OF LUTEINIZING HORMONE RELEASING HORMONE, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SYNTEX (U.S.A.) INC. (US) 1984-08-22 EP disclosed
EP-0042753-B1 NONAPEPTIDE AND DECAPEPTIDE AGONISTS OF LUTEINIZING HORMONE RELEASING HORMONE CONTAINING HETEROCYCLIC AMINO ACID RESIDUES, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOUNDS CONTAINING THEM, AND THEIR PHARMACEUTICAL USE SYNTEX (U.S.A.) INC. (US) 1984-03-21 EP disclosed
US-4338305-A LUTEINIZING HORMONE RELEASING HORMONE; CONTRACEPTIVES AMERICAN HOME PRODUCTS CORPORATION (US) 1982-07-06 US disclosed
US-4318905-A Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues SYNTEX (U.S.A.) INC. (US) 1982-03-09 US disclosed
EP-0042753-A1 Nonapeptide and decapeptide agonists of luteinizing hormone releasing hormone containing heterocyclic amino acid residues, methods for their preparation, pharmaceutical compounds containing them, and their pharmaceutical use SYNTEX (U.S.A.) INC. (US) 1981-12-30 EP disclosed
EP-0021234-A1 Nonapeptide and decapeptide derivatives of luteinizing hormone releasing hormone, their preparation and pharmaceutical compositions containing them SYNTEX (U.S.A.) INC. (US) 1981-01-07 EP disclosed
US-4234571-A CONTRACEPTIVES, ANTIFERTILITY AGENTS SYNTEX (U.S.A.) INC. (US) 1980-11-18 US disclosed