SCHEMBL4685705

SCHEMBL4685705

[CH2]CCC(=O)C1CCCN1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
PRCP P42785 2/20 0.39
DPP4 P27487 6/20 0.39
DPP8 Q6V1X1 4/20 0.38
DPP9 Q86TI2 4/20 0.38
DPP7 Q9UHL4 2/20 0.37
FAP Q12884 1/20 0.37
GLI1 P08151 1/20 0.34
MEN1 O00255 1/20 0.34
BLM P54132 1/20 0.34
KMT2A Q03164 1/20 0.34
SCN4A P35499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9579301 0.87 PRCP (0.40) NOS2NOS3NOS1PRCPDPP4
SCHEMBL9579255 0.85
SCHEMBL2645121 0.80 PRCP (0.50) NOS2NOS3NOS1PRCPDPP4
SCHEMBL30973638 0.80 PRCP (0.50) NOS2NOS3NOS1PRCPDPP4
SCHEMBL1969954 0.80 NOS2 (0.45) NOS2NOS3NOS1PRCPDPP4
SCHEMBL7432758 0.78 NOS2 (0.48) NOS2NOS3NOS1PRCPDPP4
SCHEMBL26915352 0.77 SLC22A6 (0.41) NOS2NOS3NOS1PRCPDPP4
SCHEMBL26915355 0.77 SLC22A6 (0.41) NOS2NOS3NOS1PRCPDPP4
SCHEMBL887204 0.77
SCHEMBL17929302 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed