SCHEMBL1970759

SCHEMBL1970759

CCOC(=O)C(C(N)=O)c1c[nH]c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.53
KMT2A Q03164 4/20 0.53
GPR84 Q9NQS5 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
FFAR1 O14842 2/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HTR2B P41595 1/20 0.49
MAPT P10636 4/20 0.47
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
MEN1 O00255 3/20 0.46
MGAM O43451 2/20 0.46
GAA P10253 2/20 0.46
SI P14410 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9584209 0.84 PKM (0.55) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL6190684 0.83 PKM (0.56) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL6287075 0.83 KMT2A (0.58) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL6287071 0.83 PKM (0.56) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL31458574 0.83 PKM (0.56) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL28034598 0.82 PKM (0.55) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL27836199 0.82 PKM (0.55) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL2404630 0.82 HTR4 (0.43) PKMKMT2AGPR84SMN1; SMN2FFAR1
SCHEMBL21176844 0.81 PKM (0.49) PKMKMT2AGPR84SMN1; SMN2CYP1A2
SCHEMBL14542028 0.81 HTR2A (0.54) PKMKMT2AGPR84SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334643-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES Actelion Pharmaceuticals Ltd. (CH) 2011-06-22 EP disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed