SCHEMBL19712422

SCHEMBL19712422

CCCc1nc(N2CCOCC2)cc(C)c1OC(=O)NCc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.47
ENPP2 Q13822 1/20 0.43
NAPEPLD Q6IQ20 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
USP2 O75604 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MCHR1 Q99705 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
PIK3CB P42338 2/20 0.39
PIK3CD O00329 1/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19712378 0.91 KMT2A (0.44) NAPEPLDKMT2ARAB9AKDM4EALDH1A1
SCHEMBL19712446 0.90 PPARG (0.42) THRBNAPEPLDMEN1KMT2ANPC1
SCHEMBL19712445 0.87 PIK3CA (0.42) THRBENPP2MEN1KMT2APIK3CD
SCHEMBL19712441 0.86 PIK3CA (0.40) NAPEPLDNPC1RAB9AKDM4EALDH1A1
SCHEMBL19712450 0.86 THRB (0.47) THRBENPP2NAPEPLDMEN1KMT2A
SCHEMBL19712423 0.85 SRC (0.46) NAPEPLDPIK3CBPIK3CDPIK3CA
SCHEMBL19712380 0.85 THRB (0.46) THRBENPP2NAPEPLDMEN1KMT2A
SCHEMBL2128777 0.84 MEN1 (0.51) THRBENPP2NAPEPLDMEN1KMT2A
SCHEMBL19712432 0.84 THRB (0.45) THRBENPP2NAPEPLDKDM4EALDH1A1
SCHEMBL19712372 0.84 THRB (0.44) THRBENPP2NAPEPLDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630123-B1 SUBSTITUTED 6-AMINO-NICOTINAMIDES AS KCNQ2/3 MODULATORS GRUENENTHAL GMBH (DE) 2017-12-20 EP claimed