SCHEMBL19712445

SCHEMBL19712445

CCCc1nc(N2CCOC[C@H]2C)cc(C)c1OC(=O)NCc1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.42
PIK3CD O00329 3/20 0.42
MTOR P42345 5/20 0.39
ENPP2 Q13822 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
THRB P10828 1/20 0.38
MDM2 Q00987 1/20 0.37
ATR Q13535 1/20 0.37
HTR1A P08908 1/20 0.37
GABRA1 P14867 1/20 0.37
NUDT1 P36639 1/20 0.37
RAF1 P04049 2/20 0.36
BRAF P15056 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19712400 0.92 PIK3CD (0.42) PIK3CAPIK3CDMTORKMT2AATR
SCHEMBL19712421 0.88 MTOR (0.40) PIK3CAPIK3CDMTORENPP2MEN1
SCHEMBL19712422 0.87 THRB (0.47) PIK3CAPIK3CDENPP2MEN1KMT2A
SCHEMBL19712444 0.86 MDM2 (0.42) PIK3CAPIK3CDMTORENPP2MEN1
SCHEMBL2129094 0.86 MEN1 (0.47) PIK3CAPIK3CDMTORENPP2MEN1
SCHEMBL19712390 0.81 ATR (0.41) PIK3CAPIK3CDMTORATRRAF1
SCHEMBL19712399 0.80 MTOR (0.40) PIK3CAPIK3CDMTORKMT2AATR
SCHEMBL19712378 0.79 KMT2A (0.44) PIK3CAPIK3CDMTORKMT2A
SCHEMBL19712417 0.78 POLB (0.41) PIK3CAPIK3CDMTORKMT2AATR
SCHEMBL19712427 0.77 MTOR (0.38) PIK3CAPIK3CDMTORKMT2AATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630123-B1 SUBSTITUTED 6-AMINO-NICOTINAMIDES AS KCNQ2/3 MODULATORS GRUENENTHAL GMBH (DE) 2017-12-20 EP claimed