SCHEMBL19720247

SCHEMBL19720247

CC(C)(C)OC(=O)NC(Cc1cc(O[Si](C)(C)C(C)(C)C)ccc1I)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.41
CTSS P25774 9/20 0.40
CTSK P43235 8/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
TACR1 P25103 2/20 0.39
ACE P12821 1/20 0.38
PTPN1 P18031 1/20 0.38
KLK5 Q9Y337 1/20 0.37
KDM4E B2RXH2 2/20 0.37
GLA P06280 2/20 0.37
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CTSB P07858 3/20 0.37
CTSL P07711 1/20 0.36
HPGD P15428 1/20 0.36
CACNA1B Q00975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19696953 1.00 SCN9A (0.41) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL19696793 0.88 CACNA1B (0.44) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL18788876 0.86 SCN9A (0.43) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL18788875 0.86 SCN9A (0.43) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL15856095 0.85 ITGB3 (0.43) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL19696788 0.83 CNR2 (0.41) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL15962607 0.83 ITGB3 (0.43) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL15856091 0.83 ITGB3 (0.43) SCN9ACTSSCTSKITGB3ITGA2B
SCHEMBL15856090 0.83 CTSS (0.46) SCN9ACTSSCTSKTACR1ACE
SCHEMBL15856088 0.83 CTSS (0.46) SCN9ACTSSCTSKTACR1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2940007-B1 TYROSINE DERIVATIVE AND MANUFACTURING METHOD FOR TYROSINE DERIVATIVE NARD INSTITUTE LTD (JP) 2017-12-20 EP disclosed