SCHEMBL19720609

SCHEMBL19720609

O=NC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.67
SRD5A2 P31213 1/20 0.56
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
LMNA P02545 2/20 0.53
NPSR1 Q6W5P4 1/20 0.53
P2RX1 P51575 1/20 0.53
MAPK1 P28482 1/20 0.52
POLB P06746 2/20 0.51
HPGD P15428 1/20 0.51
ALDH1A1 P00352 2/20 0.50
MAOB P27338 1/20 0.50
MAPT P10636 1/20 0.50
KCNK3 O14649 1/20 0.50
PTGS1 P23219 1/20 0.49
CNR2 P34972 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689909 0.84 CES2 (0.65) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL8504114 0.81 MAPK1 (0.63) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL6998773 0.81 CES2 (0.61) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL3176325 0.80 CES2 (1.00) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL1237189 0.80 SRD5A2 (0.79) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL5824828 0.80 CES2 (0.59) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL17664303 0.80 CES2 (0.59) CES2SRD5A2MEN1KMT2ALMNA
Hydrochloric Acid SCHEMBL7827433 0.80 MAPK1 (0.61) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL31406174 0.79 CES2 (0.69) CES2SRD5A2MEN1KMT2ALMNA
SCHEMBL9200320 0.79 CES2 (0.69) CES2SRD5A2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3257848-A1 COMPOUNDS AND COMPOSITIONS FOR MODULATING EGFR ACTIVITY Novartis AG (CH) 2017-12-20 EP disclosed