SCHEMBL8689909

SCHEMBL8689909

C[N]C(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.65
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
NPSR1 Q6W5P4 1/20 0.55
SRD5A2 P31213 1/20 0.54
ALDH1A1 P00352 2/20 0.53
POLB P06746 2/20 0.53
LMNA P02545 2/20 0.51
P2RX1 P51575 1/20 0.51
MAPK1 P28482 1/20 0.51
TP53BP1 Q12888 1/20 0.50
GAA P10253 1/20 0.50
CNR2 P34972 1/20 0.50
HTT P42858 1/20 0.50
RAB9A P51151 1/20 0.50
HPGD P15428 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
KCNK3 O14649 1/20 0.49
KCNK9 Q9NPC2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19720609 0.84 CES2 (0.67) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL4947449 0.81 CES2 (0.59) CES2MEN1KMT2AP2RX1GAA
SCHEMBL39834 0.79 CES2 (0.71) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL30093723 0.79 CES2 (0.71) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL8504114 0.79 MAPK1 (0.63) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL6998773 0.79 CES2 (0.61) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL3176325 0.79 CES2 (1.00) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL1237189 0.79 SRD5A2 (0.79) CES2MEN1KMT2ANPSR1SRD5A2
SCHEMBL20870672 0.79 CES2 (0.65) CES2MEN1KMT2ANPSR1SRD5A2
Hydrochloric Acid SCHEMBL7827433 0.78 MAPK1 (0.61) CES2MEN1KMT2ANPSR1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5795899-A Soluble salts of 4-amino-2-(4,4-dimethylimidazolidin-2-on-1-yl) pyrimidine-5-carboxylic acid N-methyl-N-(3-trifluoromethylphenyl)-amide, a process for the preparation thereof, the use thereof as pharmaceuticals and starting materials HOECHST AKTIENGESELLSCHAFT (DE) 1998-08-18 US disclosed