SCHEMBL19723014

SCHEMBL19723014

COc1ccc2nc(N)nc(C=O)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
APP P05067 1/20 0.46
KDM4E B2RXH2 3/20 0.46
POLB P06746 2/20 0.46
HSD17B10 Q99714 2/20 0.46
LMNA P02545 1/20 0.46
TRIM24 O15164 1/20 0.45
TYR P14679 1/20 0.45
TRIM33 Q9UPN9 1/20 0.45
BCHE P06276 3/20 0.45
ACHE P22303 3/20 0.45
ADORA2A P29274 2/20 0.45
CHRM1 P11229 1/20 0.45
NQO2 P16083 1/20 0.44
HPGD P15428 1/20 0.44
NCF1 P14598 1/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44
TYMS P04818 1/20 0.44
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23009237 0.78 KDM4E (0.59) ALDH1A1APPKDM4EPOLBHSD17B10
SCHEMBL15502284 0.76 NPC1 (0.51) ALDH1A1APPKDM4EPOLBHSD17B10
SCHEMBL2020170 0.75 KDM4E (0.54) ALDH1A1KDM4EPOLBHSD17B10LMNA
SCHEMBL2024081 0.75 KDM4E (0.54) ALDH1A1KDM4EPOLBHSD17B10LMNA
SCHEMBL1876646 0.73 ADORA2A (0.51) ALDH1A1APPKDM4EBCHEACHE
SCHEMBL28910000 0.72 POLB (0.61) ALDH1A1KDM4EPOLBHSD17B10LMNA
SCHEMBL28026104 0.72 POLB (0.59) ALDH1A1KDM4EPOLBHSD17B10LMNA
SCHEMBL27787446 0.72 DCPS (0.57) ALDH1A1APPKDM4EPOLBHSD17B10
SCHEMBL12637539 0.71 TRIM24 (0.54) ALDH1A1KDM4EPOLBHSD17B10LMNA
SCHEMBL12637535 0.71 TRIM24 (0.54) ALDH1A1KDM4EPOLBHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709989-B1 QUINAZOLINE DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS AND FURTHER DISEASES JANSSEN SCIENCES IRELAND UC (IE) 2017-12-20 EP disclosed