SCHEMBL19730136

SCHEMBL19730136

CNc1nccc2c1c(/C=C/C(=O)OC)nn2Cc1ccc(OC)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
CCR4 P51679 1/20 0.38
PTGER4 P35408 2/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
BUB1 O43683 2/20 0.35
CSF1R P07333 1/20 0.35
ALOX15 P16050 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
HDAC5 Q9UQL6 2/20 0.34
HSP90AA1 P07900 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31500887 1.00 JAK2 (0.39) JAK2CCR4PTGER4CNR1CNR2
SCHEMBL21434366 0.92 JAK2 (0.39) JAK2CCR4PTGER4CNR1CNR2
SCHEMBL3775379 0.88 CCR4 (0.39) JAK2CCR4PTGER4CNR1CNR2
SCHEMBL3775383 0.88 CCR4 (0.39) JAK2CCR4PTGER4CNR1CNR2
SCHEMBL416412 0.86 JAK2 (0.48) JAK2L3MBTL1ALDH1A1LMNAPOLB
SCHEMBL416411 0.86 JAK2 (0.48) JAK2L3MBTL1ALDH1A1LMNAPOLB
SCHEMBL10225762 0.84 JAK2 (0.47) JAK2CCR4L3MBTL1ALDH1A1POLB
SCHEMBL3771429 0.79 CNR1 (0.41) PTGER4CNR1CNR2BUB1L3MBTL1
SCHEMBL3772381 0.79 CNR1 (0.41) PTGER4CNR1CNR2BUB1L3MBTL1
SCHEMBL19730053 0.78 CNR1 (0.43) JAK2CCR4PTGER4CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017215600-A1 SUBSTITUTED TRICYCLIC HERTEOCYCLIC COMPOUNDS AND USE THEREOF SUZHOU YABAO PHARMACEUTICAL R&D CO., LTD. (CN) 2017-12-21 WO disclosed