SCHEMBL19734472

SCHEMBL19734472

CCC(OC)c1ccc(Br)cc1C#N

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.34
MAOA P21397 2/20 0.34
AAK1 Q2M2I8 2/20 0.33
EGFR P00533 3/20 0.32
ERBB2 P04626 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
APLNR P35414 2/20 0.31
TSHR P16473 2/20 0.31
HPGD P15428 1/20 0.31
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469317 0.83 APLNR (0.36) SMN1; SMN2APLNRTSHRHPGD
SCHEMBL19713336 0.80 KDM4E (0.39) MAOBMAOAAAK1EGFRERBB2
SCHEMBL24767628 0.79 SMN1; SMN2 (0.36) MAOBMAOAAAK1EGFRERBB2
SCHEMBL12251161 0.74 GABRA1 (0.42) MAOBMAOAAAK1SMN1; SMN2NOS3
SCHEMBL18638444 0.73 SMN1; SMN2 (0.34) MAOBMAOAAAK1SMN1; SMN2NOS3
SCHEMBL27945351 0.73 MAOB (0.37) MAOBMAOAAAK1SMN1; SMN2NOS3
SCHEMBL24416900 0.72 MAOB (0.39) MAOBMAOAAAK1SMN1; SMN2NOS3
SCHEMBL1780515 0.71 MAOB (0.38) MAOBMAOAAAK1SMN1; SMN2NOS3
SCHEMBL392560 0.70 MAOB (0.47) MAOBMAOAAAK1EGFRERBB2
SCHEMBL22904500 0.70 KMT2A (0.45) AAK1EGFRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216280-A1 TETRAHYDRO-PYRIDO[3,4-b]INDOLE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-12-21 WO disclosed