SCHEMBL19734568

SCHEMBL19734568

CCc1c(C#N)c(C)nc(N2CCCN(C)CC2)c1C#N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.44
ALDH1A1 P00352 7/20 0.44
HPGD P15428 5/20 0.44
GAA P10253 1/20 0.44
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 3/20 0.41
POLB P06746 2/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
ADRA2A P08913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19734810 0.95 CYP2C19 (0.45) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL19717348 0.86 KDM4E (0.43) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL30995100 0.86 ALDH1A1 (0.43) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL30995087 0.86 KDM4E (0.51) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL19734567 0.80 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10KMT2A
SCHEMBL19739015 0.78 ALDH1A1 (0.47) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL19734951 0.77 DNMT1 (0.44) KDM4EALDH1A1HPGDGAARECQL
SCHEMBL29658540 0.77 KDM4E (0.43) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL29658799 0.77 KDM4E (0.43) KDM4EALDH1A1HPGDGAAKMT2A
SCHEMBL19716884 0.76 ALDH1A1 (0.47) KDM4EALDH1A1HPGDGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed