SCHEMBL19734567

SCHEMBL19734567

CCc1c(C#N)c(C)nc(N2CCOCC2)c1C#N

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 14/20 0.55
ALDH1A1 P00352 14/20 0.55
POLB P06746 1/20 0.55
HPGD P15428 9/20 0.55
KHK P50053 1/20 0.55
NUDT1 P36639 1/20 0.52
HSD17B10 Q99714 4/20 0.50
HTT P42858 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ATM Q13315 2/20 0.48
LMNA P02545 5/20 0.46
TSHR P16473 2/20 0.46
MAPK1 P28482 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29658476 0.84 KDM4E (0.54) KDM4EALDH1A1POLBHPGDKHK
SCHEMBL19734698 0.84 KDM4E (0.54) KDM4EALDH1A1POLBHPGDKHK
SCHEMBL19717161 0.84 KDM4E (0.54) KDM4EALDH1A1POLBHPGDKHK
SCHEMBL19734810 0.84 CYP2C19 (0.45) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL19734951 0.81 DNMT1 (0.44) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL19734568 0.80 KDM4E (0.44) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL19734298 0.74 KDM5A (0.45) KDM4EALDH1A1POLBHPGDHSD17B10
SCHEMBL30762361 0.72 ALDH1A1 (0.49) KDM4EALDH1A1POLBHPGDKHK
SCHEMBL30762379 0.71 ALDH1A1 (0.48) KDM4EALDH1A1POLBHPGDKHK
SCHEMBL17344002 0.71 ALDH1A1 (1.00) KDM4EALDH1A1POLBHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed