SCHEMBL19734735

SCHEMBL19734735

Cc1c(C#N)c(O)nc(O)c1C#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
GAA P10253 3/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
HTT P42858 2/20 0.35
GLA P06280 1/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 7/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33
UPP1 Q16831 2/20 0.32
ADRA2A P08913 1/20 0.32
ADORA2A P29274 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RECQL P46063 1/20 0.31
MAPT P10636 1/20 0.31
CACNA1B Q00975 1/20 0.31
APBA1 Q02410 1/20 0.31
CDK4 P11802 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7238065 0.90 ALDH1A1 (0.36) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL28686642 0.84 HTT (0.46) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL30692217 0.84 HTT (0.46) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL21686185 0.81 ALDH1A1 (0.38) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL10728519 0.80 KDM4E (0.44) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL4673214 0.78 HTT (0.58) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL11100290 0.78 KMT2A (0.44) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL8650240 0.78 ATM (0.39) ALDH1A1GAAHPGDMEN1KMT2A
SCHEMBL11826533 0.77 ALDH1A1 (0.37) ALDH1A1GAAHPGDKDM4EADORA2A
SCHEMBL19716478 0.77 MAPT (0.40) ALDH1A1GAAHPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216727-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed
WO-2017216726-A1 SUBSTITUTED PYRIDINES AS INHIBITORS OF DNMT1 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-12-21 WO disclosed