SCHEMBL1975972

SCHEMBL1975972

CC1(CNC(=O)OCc2ccccc2)CCCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 3/20 0.39
GSK3B P49841 7/20 0.39
CYP2D6 P10635 3/20 0.39
MAP4K1 Q92918 1/20 0.37
TSHR P16473 2/20 0.37
FSHR P23945 2/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
GRIN2B Q13224 1/20 0.36
GAA P10253 1/20 0.35
POLB P06746 1/20 0.35
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CYP46A1 Q9Y6A2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1975690 0.79 CYP2D6 (0.42) FKBP1AGSK3BCYP2D6CYP3A4CYP2C9
SCHEMBL1831688 0.78 CYP2D6 (0.42) GSK3BCYP2D6CYP3A4CYP2C9GRIN2B
SCHEMBL15512999 0.77 GSK3B (0.44) GSK3BCYP2D6
SCHEMBL1832408 0.77 GSK3B (0.42) GSK3BCYP2D6CYP46A1
SCHEMBL3273975 0.73 GSK3B (0.47) GSK3BCYP2D6POLB
SCHEMBL2066100 0.70 GSK3B (0.43) GSK3BCYP2D6CYP3A4
SCHEMBL3278253 0.70 ATM (0.45) GSK3BCYP2D6POLB
SCHEMBL3280949 0.70 GSK3B (0.45) GSK3BCYP2D6POLB
SCHEMBL4385699 0.68 GSK3B (0.35) GSK3BCYP2D6CYP3A4
SCHEMBL4387999 0.68 GSK3B (0.37) GSK3BTSHRCYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110144132-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES SANOFI-AVENTIS (FR) 2011-06-16 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110144132-A1 SUBSTITUTED PYRIMIDIN-4-ONE DERIVATIVES TYMP, DHFR, DPYD FKBP1A 3961/4885GSK3B 3574/4885CYP2D6 221/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.