SCHEMBL4385699

SCHEMBL4385699

CC1(NC(=O)c2ccc3ncccc3n2)CCCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.35
NAMPT P43490 1/20 0.34
CYP3A4 P08684 4/20 0.34
LATS1 O95835 1/20 0.33
LATS2 Q9NRM7 1/20 0.33
CYP2D6 P10635 2/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4392100 0.98 GSK3B (0.35) GSK3BNAMPTCYP3A4LATS1LATS2
SCHEMBL4384554 0.83 GSK3B (0.37) GSK3BCYP3A4CYP2D6
SCHEMBL4954713 0.82 GSK3B (0.36) GSK3BCYP3A4LATS1LATS2CYP2D6
SCHEMBL4377775 0.81 GSK3B (0.39) GSK3BLATS1LATS2CYP2D6HDAC1
SCHEMBL4378591 0.80 GSK3B (0.38) GSK3BCYP3A4CYP2D6
SCHEMBL4383569 0.78 GSK3B (0.37) GSK3BCYP3A4CYP2D6
SCHEMBL2066100 0.78 GSK3B (0.43) GSK3BCYP3A4CYP2D6
SCHEMBL4387999 0.77 GSK3B (0.37) GSK3BCYP3A4
SCHEMBL4384596 0.77 GSK3B (0.37) GSK3BNAMPTCYP3A4CYP2D6
SCHEMBL3373754 0.75 OPRD1 (0.41) GSK3BCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed