SCHEMBL1978207

SCHEMBL1978207

Nc1ccc(OC2CCC2)cc1-c1cc(Cl)ncc1Cl

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.36
BTK Q06187 1/20 0.36
KDM1A O60341 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
PARP10 Q53GL7 1/20 0.35
FFAR4 Q5NUL3 2/20 0.34
ROCK1 Q13464 3/20 0.33
FURIN P09958 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
ROCK2 O75116 1/20 0.33
KCNH2 Q12809 1/20 0.33
PRKCZ Q05513 1/20 0.33
PDK2 Q15119 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12597604 0.80 FFAR4 (0.37) ABL1SLC40A1FFAR4HRH3PDK2
SCHEMBL1983238 0.78 HSP90AA1 (0.47) KDM1A
SCHEMBL19641652 0.76 SLC6A2 (0.46) PARP10FFAR4FURINHRH3PDK2
SCHEMBL1980018 0.73 KDM1A (0.34) KDM1A
SCHEMBL1980019 0.73 CHEK2 (0.40) KDM1A
SCHEMBL25956126 0.73 SLC6A2 (0.46) PARP10FFAR4HRH3PDK2SLC6A2
SCHEMBL27253444 0.71 HPGD (0.47) ABL1PARP10FFAR4HRH3PDK2
SCHEMBL17396860 0.70 LOX (0.40) ABL1SLC40A1PARP10ROCK1ROCK2
SCHEMBL13875187 0.69 ABL1 (0.53) ABL1ROCK1ROCK2KCNH2PRKCZ
SCHEMBL1981906 0.68 GABRA1 (0.52) ABL1SLC40A1ROCK1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed