SCHEMBL19782657

SCHEMBL19782657

CC(C)(C)[Si](C)(C)OCc1cc(N)ccc1C=O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.39
TRIM24 O15164 1/20 0.31
TYR P14679 1/20 0.31
TRIM33 Q9UPN9 1/20 0.31
ELANE P08246 1/20 0.30
TACR1 P25103 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17494744 0.84 TDP1 (0.41) BACE1TRIM24TYRTRIM33
SCHEMBL30219107 0.80 BACE1 (0.56) BACE1TRIM24TRIM33TACR1
SCHEMBL2082920 0.80 BACE1 (0.56) BACE1TRIM24TRIM33TACR1
SCHEMBL18149538 0.79 CYP3A4 (0.37) BACE1
SCHEMBL25284529 0.79 BACE1 (0.36) BACE1
SCHEMBL21163340 0.78 ALDH1A1 (0.39) BACE1
SCHEMBL9125186 0.78 BACE1 (0.38) BACE1
SCHEMBL23462893 0.78 IDO1 (0.44) BACE1
SCHEMBL16880571 0.77 BACE1 (0.39) BACE1TACR1
SCHEMBL18071006 0.77 GAA (0.39) BACE1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190292176-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BISTOL MYERS SQUIBB COMPANY (US) 2019-09-26 US disclosed
WO-2018013774-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-01-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190292176-A1 BICYCLIC HETEROARYL SUBSTITUTED COMPOUNDS F2, F2RL3, PF4 BACE1 1192/4885TRIM24 4734/4885TYR 477/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.