SCHEMBL1978484

SCHEMBL1978484

COC(C)Oc1ccc2[nH]c3cnc(-c4cnn(C)c4)cc3c2c1-c1ccc(C(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.42
PIM1 P11309 6/20 0.40
MAP4K4 O95819 1/20 0.39
ACHE P22303 1/20 0.37
PIM3 Q86V86 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
PLAU P00749 1/20 0.36
MAP4K1 Q92918 1/20 0.36
MAPT P10636 1/20 0.36
HAT1 O14929 2/20 0.36
EP300 Q09472 2/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
TTK P33981 1/20 0.36
GSK3B P49841 2/20 0.35
DYRK1A Q13627 2/20 0.35
TLR8 Q9NR97 1/20 0.35
TLR7 Q9NYK1 1/20 0.35
FLT3 P36888 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1982173 0.91 CHEK1 (0.45) CHEK1PIM1MAP4K4ACHEPIM3
SCHEMBL12597208 0.87 CHEK1 (0.42) CHEK1PIM1MAP4K4ACHEPIM3
SCHEMBL1983422 0.86 CHEK1 (0.42) CHEK1PIM1MAP4K4ACHEPIM3
SCHEMBL1983392 0.81 PIM1 (0.45) CHEK1PIM1ACHEPIM3PIM2
SCHEMBL1982365 0.80 NEK1 (0.39) CHEK1PIM1ACHEPIM3PIM2
SCHEMBL1984109 0.78 CHEK1 (0.48) CHEK1PIM1MAP4K4ACHEPIM3
SCHEMBL12597220 0.77 TLR7 (0.41) MAP4K1CCNA2CDK2TTKTLR8
SCHEMBL11908677 0.77 CHEK1 (0.47) CHEK1PIM1MAP4K4ACHEPIM3
SCHEMBL1979521 0.77 PIM1 (0.50) CHEK1PIM1ACHEPIM3PIM2
SCHEMBL12597221 0.75 GSK3B (0.40) CHEK1PIM1PLAUMAP4K1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed