SCHEMBL19785779

SCHEMBL19785779

CC(=O)c1cc(C)cc([N+](=O)[O-])c1C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.55
TSHR P16473 4/20 0.46
CYP3A4 P08684 1/20 0.46
CYP1A2 P05177 1/20 0.42
DHODH Q02127 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6830067 0.85 TSHR (0.59) GPR35TSHRCYP3A4CYP1A2KDM4E
SCHEMBL31392530 0.84 GPR35 (0.69) GPR35TSHRCYP3A4CYP1A2KDM4E
SCHEMBL4132017 0.84 GPR35 (0.69) GPR35TSHRCYP3A4CYP1A2KDM4E
SCHEMBL13468191 0.82 DHODH (0.52) TSHRDHODHALDH1A1MEN1KMT2A
SCHEMBL31399740 0.82 TSHR (0.44) GPR35TSHRCYP1A2DHODHMAPT
SCHEMBL13468174 0.82 CYP1A2 (0.47) GPR35TSHRCYP1A2DHODHMAPT
SCHEMBL6828146 0.82 GPR35 (0.52) GPR35TSHRCYP3A4MAPTALDH1A1
SCHEMBL28051861 0.80 GPR35 (0.49) GPR35TSHRCYP3A4CYP1A2MAPT
SCHEMBL260768 0.80 GPR35 (0.67) GPR35TSHRCYP3A4CYP1A2KDM4E
SCHEMBL1277039 0.78 TSHR (0.60) GPR35TSHRCYP3A4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018011201-A1 HETEROAROMATIC MODULATORS OF THE RETINOID-RELATED ORPHAN RECEPTOR GAMMA LEO PHARMA A/S (DK) 2018-01-18 WO disclosed