SCHEMBL19785898

SCHEMBL19785898

COc1cccc(SC/C=C/SSCc2ccc(C)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.46
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
MTNR1A P48039 4/20 0.38
MTNR1B P49286 4/20 0.38
CYP1A2 P05177 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C8 P10632 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
ACHE P22303 2/20 0.37
BCHE P06276 1/20 0.37
DHFR P00374 1/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21189911 0.90 MAOB (0.43) MAOBMAPTTP53POLBMTNR1A
SCHEMBL21189901 0.90 MAOB (0.43) MAOBMAPTTP53POLBMTNR1A
SCHEMBL21190028 0.89 MAOB (0.47) MAOBMTNR1AMTNR1BCYP1A2CYP3A4
SCHEMBL21190019 0.89 MAOB (0.47) MAOBMTNR1AMTNR1BCYP1A2CYP3A4
SCHEMBL21190093 0.89 ALDH1A1 (0.39) MAOBMAPTMTNR1AMTNR1BCYP1A2
SCHEMBL21189962 0.89 ALDH1A1 (0.39) MAOBMAPTMTNR1AMTNR1BCYP1A2
SCHEMBL19785872 0.88 ADORA2A (0.37) MAOBPOLBMTNR1AMTNR1BCYP1A2
SCHEMBL21190021 0.85 HRH1 (0.40) MAOBMAPTPOLBMTNR1AMTNR1B
SCHEMBL21189916 0.85 HRH1 (0.40) MAOBMAPTPOLBMTNR1AMTNR1B
SCHEMBL19785649 0.85 APP (0.47) MAOBMAPTTP53CYP1A2CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018012947-A1 NOVEL ORGANIC SULFUR COMPOUND, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER OR AN INFLAMMATORY DISEASE, CONTAINING SAME AS ACTIVE INGREDIENT 숙명여자대학교 산학협력단 2018-01-18 WO disclosed