SCHEMBL1978668

SCHEMBL1978668

CCOC(=O)c1ccc(C)c([N+](=O)[O-])c1.Cc1ccc(C(=O)O)cc1[N+](=O)[O-]

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.75
KMT2A Q03164 2/20 0.61
ALDH1A1 P00352 3/20 0.60
MAPT P10636 3/20 0.60
PKM P14618 2/20 0.60
RAB9A P51151 2/20 0.60
NPC1 O15118 1/20 0.60
CRHBP P24387 1/20 0.60
CRHR2 Q13324 1/20 0.60
KDM4E B2RXH2 2/20 0.58
LMNA P02545 1/20 0.58
POLB P06746 1/20 0.58
MEN1 O00255 1/20 0.57
AGTR1 P30556 1/20 0.57
HPGD P15428 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
PTGER4 P35408 1/20 0.56
CES2 O00748 1/20 0.56
CES1 P23141 1/20 0.56
CASP6 P55212 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981486 0.94 KMT2A (0.67) TSHRKMT2AALDH1A1MAPTPKM
SCHEMBL177231 0.87 TSHR (1.00) TSHRKMT2AALDH1A1MAPTRAB9A
SCHEMBL30668892 0.87 TSHR (1.00) TSHRKMT2AALDH1A1MAPTRAB9A
4-Chloro-3-Nitrobenzoic Acid SCHEMBL7843735 0.86 KMT2A (0.58) TSHRKMT2AALDH1A1MAPTPKM
Ammonia Solution, Strong SCHEMBL27660564 0.85 TSHR (0.96) TSHRKMT2AALDH1A1MAPTRAB9A
Hydrochloric Acid SCHEMBL11517993 0.85 TSHR (0.96) TSHRKMT2AALDH1A1MAPTRAB9A
SCHEMBL7941824 0.84 KMT2A (0.62) TSHRKMT2AALDH1A1MAPTPKM
Hydrochloric Acid SCHEMBL11776974 0.83 TSHR (0.57) TSHRKMT2AALDH1A1MAPTPKM
Hydrochloric Acid SCHEMBL11780689 0.83 KMT2A (0.61) TSHRKMT2AALDH1A1MAPTPKM
SCHEMBL5262777 0.83 KMT2A (0.55) TSHRKMT2AALDH1A1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509980-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE Boehringer Ingelheim International GmbH (DE) 2012-10-17 EP disclosed
WO-2011071716-A1 HETEROCYCLIC COMPOUNDS CONTAINING AN INDOLE CORE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-06-16 WO disclosed