SCHEMBL7941824

SCHEMBL7941824

CCOC(=O)c1ccc(C(=O)O)c([N+](=O)[O-])c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.62
ALDH1A1 P00352 5/20 0.61
MAPT P10636 2/20 0.61
RAB9A P51151 2/20 0.61
NPC1 O15118 2/20 0.61
PKM P14618 1/20 0.61
CRHBP P24387 1/20 0.61
CRHR2 Q13324 1/20 0.61
LMNA P02545 2/20 0.60
POLB P06746 2/20 0.60
KDM4E B2RXH2 1/20 0.60
PTGER4 P35408 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.53
GAA P10253 1/20 0.53
TSHR P16473 2/20 0.51
MEN1 O00255 1/20 0.51
THRB P10828 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11780689 0.99 KMT2A (0.61) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL6422578 0.91 KMT2A (0.65) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL4753200 0.89 KMT2A (0.59) KMT2AALDH1A1MAPTRAB9ANPC1
Hydrochloric Acid SCHEMBL11776974 0.87 TSHR (0.57) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL11780686 0.87 KMT2A (0.61) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL28066675 0.87 KMT2A (0.57) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL28230924 0.85 KMT2A (0.56) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL18779429 0.85 KMT2A (0.58) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL1978668 0.84 TSHR (0.75) KMT2AALDH1A1MAPTRAB9ANPC1
SCHEMBL1981486 0.84 KMT2A (0.67) KMT2AALDH1A1MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6268496-B1 GAMMA-AMINOBUTYRIC ACID RECEPTOR LIGANDS NEUROGEN CORPORATION 2001-07-31 US disclosed
EP-0555391-B1 CERTAIN IMIDAZOQUINOXALINES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORP (US) 2000-07-12 EP disclosed
US-5744602-A PSYCHOLOGICAL DISORDERS, ANTICONVULSANTS NEUROGEN CORPORATION (US) 1998-04-28 US disclosed
CN-1034174-C Certain imidazoquinoxalines, a new class of GABA brain receptor ligands NEUROGEN CORP (US) 1997-03-05 CN disclosed
CN-1076930-A Some imidazo quinoxaline compound; The γ-An Jidingsuan brain receptor ligands that one class is new NEUROGEN CORP (US) 1993-10-06 CN disclosed
EP-0555391-A1 CERTAIN IMIDAZOQUINOXALINES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1993-08-18 EP disclosed
US-5130430-A Anxiety, sleep disorders or seizures NEUROGEN CORPORATION (US) 1992-07-14 US disclosed
WO-1992007853-A1 CERTAIN IMIDAZOQUINOXALINES; A NEW CLASS OF GABA BRAIN RECEPTOR LIGANDS NEUROGEN CORPORATION (US) 1992-05-14 WO disclosed