SCHEMBL19789518

SCHEMBL19789518

C=CC(=O)OCCCOc1ccc2cc(C#Cc3ccc(N=S)cc3)ccc2c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.42
TSHR P16473 2/20 0.36
HPGD P15428 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
ACACB O00763 5/20 0.34
FFAR1 O14842 5/20 0.34
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
MTNR1A P48039 4/20 0.32
MTNR1B P49286 4/20 0.32
FURIN P09958 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12437039 0.91 THRB (0.50) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL12436997 0.90 THRB (0.41) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL16133506 0.88 THRB (0.39) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL19821125 0.86 THRB (0.52) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL14907431 0.85 THRB (0.45) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL14907509 0.85 THRB (0.45) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL12437000 0.85 THRB (0.45) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL14907503 0.84 THRB (0.46) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL14302569 0.83 THRB (0.45) THRBTSHRHPGDALDH1A1CYP3A4
SCHEMBL12437036 0.83 THRB (0.42) THRBTSHRHPGDALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2771735-B1 SWITCH ELEMENT COMPRISING A LIQUID CRYSTALLINE MEDIUM MERCK PATENT GMBH (DE) 2018-01-24 EP disclosed