SCHEMBL19789643

SCHEMBL19789643

CCc1ccc(CCC(C)(C)C)c(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
HSPA5 P11021 1/20 0.33
S1PR1 P21453 2/20 0.33
FFAR4 Q5NUL3 1/20 0.33
IDO1 P14902 4/20 0.33
PDE2A O00408 1/20 0.33
TRPA1 O75762 1/20 0.32
AOC3 Q16853 1/20 0.32
DAO P14920 1/20 0.32
PDK2 Q15119 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2A6 P11509 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12114208 0.84 S1PR1 (0.37) PDE3BPDE3AS1PR1FFAR4IDO1
SCHEMBL12834802 0.82 FFAR4 (0.40) HSPA5FFAR4IDO1TRPA1DAO
SCHEMBL23865007 0.80 ESRRG (0.41) PDE3BPDE3AHSPA5AOC3DAO
SCHEMBL24250763 0.79 S1PR1 (0.38) PDE3BPDE3AS1PR1TRPA1CYP1A2
SCHEMBL25530531 0.78 PDE3B (0.45) PDE3BPDE3AIDO1DAOCYP1A2
SCHEMBL12107918 0.75 CNR1 (0.41) S1PR1IDO1DAOPDK2
SCHEMBL3245823 0.74 RXRA (0.44) FFAR4IDO1PDE2ATRPA1DAO
SCHEMBL27408304 0.73 TP53 (0.42) PDK2CYP1A2CYP2A6SLC6A4SIGMAR1
SCHEMBL23463560 0.73 HSPA5 (0.44) HSPA5IDO1PDK2CYP1A2CYP2A6
SCHEMBL17891892 0.73 PDE3B (0.44) PDE3BPDE3AS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3272736-A1 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS NOVARTIS AG (CH) 2018-01-24 EP disclosed