SCHEMBL1978989

SCHEMBL1978989

COc1ccc(N)c(-c2cc(-c3cccnc3)ncc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
RAB9A P51151 2/20 0.58
CYP11B2 P19099 7/20 0.49
CYP11B1 P15538 6/20 0.49
CYP17A1 P05093 4/20 0.49
CYP3A4 P08684 4/20 0.49
KDM4E B2RXH2 6/20 0.48
NPSR1 Q6W5P4 3/20 0.48
CYP19A1 P11511 2/20 0.47
RXFP1 Q9HBX9 2/20 0.46
CYP1A2 P05177 3/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1B1 Q16678 1/20 0.46
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP2D6 P10635 2/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
GLA P06280 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12594806 0.85 CHRM5 (0.48) NPC1RAB9ACYP11B2CYP11B1
SCHEMBL12594726 0.81 KDM4E (0.44) NPC1RAB9ACYP11B2CYP11B1CYP3A4
SCHEMBL12594372 0.79 PIM1 (0.47) NPC1RAB9ACYP11B2CYP11B1CYP19A1
SCHEMBL1983238 0.78 HSP90AA1 (0.47) NPC1RAB9ACYP11B2CYP11B1CYP3A4
SCHEMBL1981896 0.78 NPC1 (0.45) NPC1RAB9ACYP11B2CYP11B1CYP17A1
SCHEMBL473704 0.76 ADORA2A (0.45) NPC1RAB9ACYP3A4KDM4EALDH1A1
SCHEMBL1561017 0.74 CHEK2 (0.44) NPC1RAB9ACYP3A4ATR
SCHEMBL473747 0.72 JAK2 (0.44) KDM4EALDH1A1HPGDGLAATR
SCHEMBL1560831 0.71 PDE4A (0.42) RAB9ACYP11B2CYP11B1CYP3A4CYP19A1
SCHEMBL12435508 0.70 CYP2A6 (0.58) NPC1RAB9ACYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed