SCHEMBL1979009

SCHEMBL1979009

COc1ccc2[nH]c3cnc(-c4cccnc4)cc3c2c1-c1ccc(C(=O)NC2CCNC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.46
DYRK1A Q13627 6/20 0.44
WNT1 P04628 5/20 0.44
DGAT2 Q96PD7 4/20 0.42
PDPK1 O15530 1/20 0.41
SUV39H2 Q9H5I1 2/20 0.41
NRAS P01111 1/20 0.40
LCK P06239 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
FLT3 P36888 1/20 0.40
CDK7 P50613 1/20 0.40
IRAK1 P51617 1/20 0.40
CCNH P51946 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
CHEK2 O96017 1/20 0.40
MET P08581 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12597832 0.92 DYRK1A (0.45) PIM1DYRK1AWNT1
SCHEMBL1978545 0.88 IGF1R (0.41) PIM1DYRK1AWNT1
SCHEMBL12597625 0.87 IGF1R (0.43) PIM1DYRK1AWNT1
SCHEMBL12598118 0.84
SCHEMBL12597359 0.83 SLC2A1 (0.45) PIM1
SCHEMBL1983761 0.83 BRAF (0.47) PIM1DYRK1AWNT1
SCHEMBL1981803 0.82 MTNR1A (0.45) PIM1
SCHEMBL1980514 0.82 PIM1 (0.44) PIM1DYRK1A
SCHEMBL1980453 0.82 SUV39H2 (0.43) SUV39H2CHEK2MET
SCHEMBL1981315 0.82 PTAFR (0.47) DYRK1AWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070299-A1 TRI-SUBSTITUTED 9H-BETA-CARBOLINE (OR 9H-PYRIDO[3,4-B]INDOLE) DERIVATIVES, PREPARATION OF SAME AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-06-16 WO disclosed