SCHEMBL19790355

SCHEMBL19790355

C=C(CC(C)(C)C)N[C@@H](C)C(C)Nc1nc(N)c(C#N)cc1F

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HTT P42858 1/20 0.33
KHK P50053 1/20 0.33
IRAK4 Q9NWZ3 10/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
JAK2 O60674 1/20 0.30
JAK3 P52333 1/20 0.30
LIMK1 P53667 1/20 0.30
LIMK2 P53671 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19790349 0.83
SCHEMBL19790110 0.78 JAK3 (0.34) KDM4EMAPTJAK2JAK3LIMK1
SCHEMBL19790864 0.76
SCHEMBL19790695 0.76 JAK2 (0.38) KDM4EALDH1A1IRAK4RAB9AJAK2
SCHEMBL19790790 0.70
SCHEMBL7859690 0.70 KHK (0.45) KDM4EALDH1A1LMNAHSD17B10HTT
SCHEMBL19790715 0.68
SCHEMBL19790398 0.68
SCHEMBL19790125 0.68
SCHEMBL19790549 0.67 SYK (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2799431-B1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORP (JP) 2018-01-24 EP disclosed