SCHEMBL19790695

SCHEMBL19790695

C=C(CC(C)(C)C)N[C@@H](C)C(C)Nc1nc(Nc2ccc3ncccc3c2)c(C#N)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
IRAK4 Q9NWZ3 2/20 0.37
SYK P43405 1/20 0.37
GRM4 Q14833 2/20 0.36
ALDH1A1 P00352 3/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
EGFR P00533 2/20 0.33
POLB P06746 2/20 0.33
BRAF P15056 1/20 0.33
TNF P01375 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19790420 0.85 SYK (0.51) IRAK4SYKALDH1A1NPC1RAB9A
SCHEMBL14929079 0.84 TRPA1 (0.40) JAK2JAK1IRAK4SYKGRM4
SCHEMBL14910328 0.82 GRM4 (0.42) JAK2JAK1SYKGRM4ALDH1A1
SCHEMBL14928547 0.82 GRM4 (0.42) JAK2JAK1SYKGRM4ALDH1A1
SCHEMBL14929941 0.80 HPGD (0.46) JAK2JAK1SYKGRM4ALDH1A1
SCHEMBL19790110 0.79 JAK3 (0.34) JAK2KDM4E
SCHEMBL14910387 0.79 GRM4 (0.41) JAK2JAK1SYKGRM4ALDH1A1
SCHEMBL14910389 0.79 GRM4 (0.41) JAK2JAK1SYKGRM4ALDH1A1
SCHEMBL14910413 0.79 IRAK4 (0.37) JAK2JAK1IRAK4SYKGRM4
SCHEMBL14928328 0.79 HPGD (0.44) JAK2JAK1SYKGRM4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2799431-B1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORP (JP) 2018-01-24 EP disclosed