SCHEMBL1979148

SCHEMBL1979148

Oc1ccc(-c2cc[c]cc2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.43
AR P10275 4/20 0.42
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
USP7 Q93009 2/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
ESR1 P03372 5/20 0.35
ESR2 Q92731 4/20 0.35
APP P05067 1/20 0.33
PGR P06401 1/20 0.33
ABL1 P00519 1/20 0.32
ABCB1 P08183 1/20 0.32
BCR P11274 1/20 0.32
TNIK Q9UKE5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636363 0.84 KIF11 (0.41) KIF11ARAPP
SCHEMBL2433534 0.84 PDE3B (0.36) KIF11ARPDE3BPDE3APGR
SCHEMBL6513960 0.82 PDE3B (0.37) ARPDE3BPDE3A
SCHEMBL1369645 0.81 KIF11 (0.38) KIF11AR
SCHEMBL9586467 0.81 APP (0.43) KIF11ARHSD17B1HSD17B2APP
SCHEMBL14483362 0.80 GLA (0.38)
SCHEMBL8821891 0.79 KIF11 (0.42) KIF11PDE3BPDE3A
SCHEMBL7955020 0.78 PGR (0.47) ARESR2PGRABL1ABCB1
SCHEMBL2431534 0.76 PDE3B (0.40) KIF11ARPDE3BPDE3A
SCHEMBL4669684 0.76 AKR1C3 (0.48) KIF11ARAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509978-A1 AZOCYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE E.I. Du Pont De Nemours And Company (US) 2012-10-17 EP disclosed
WO-2011072207-A1 AZOCYCLIC INHIBITORS OF FATTY ACID AMIDE HYDROLASE E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-06-16 WO disclosed