SCHEMBL19795013

SCHEMBL19795013

COc1nn(-c2cnc(C(F)(F)F)nc2)cc1C=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 8/20 0.40
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
NLRP3 Q96P20 1/20 0.38
PTGS2 P35354 2/20 0.34
POLB P06746 2/20 0.32
ALDH1A1 P00352 2/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
KDM4E B2RXH2 1/20 0.30
THRB P10828 1/20 0.30
PKM P14618 1/20 0.30
RECQL P46063 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16648002 0.84 TRPA1 (0.45) TRPA1KMT2AMEN1NLRP3PTGS2
SCHEMBL16635554 0.81 KMT2A (0.43) TRPA1KMT2AMEN1NLRP3PTGS2
SCHEMBL17979498 0.80 TRPA1 (0.40) TRPA1
SCHEMBL19795019 0.80 PTGS2 (0.37) TRPA1KMT2AMEN1NLRP3PTGS2
SCHEMBL16635488 0.77 TRPA1 (0.43) TRPA1KMT2AMEN1POLBALDH1A1
SCHEMBL17973850 0.77 TRPA1 (0.43) TRPA1KMT2AALDH1A1
SCHEMBL28847111 0.76 TRPA1 (0.41) TRPA1
SCHEMBL717945 0.76 MEN1 (0.47) KMT2AMEN1NLRP3PTGS2POLB
SCHEMBL16635561 0.76 TRPA1 (0.43) TRPA1KMT2AALDH1A1KDM4EPKM
SCHEMBL16647990 0.75 TRPA1 (0.46) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3487853-B1 BICYCLIC PROLINE COMPOUNDS HOFFMANN LA ROCHE (CH) 2022-06-08 EP disclosed
WO-2018015410-A1 BICYCLIC PROLINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2018-01-25 WO disclosed