SCHEMBL1979528

SCHEMBL1979528

CCCCN(Cc1ccccc1F)c1nnc(-c2ccnc(O)c2)s1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.44
S1PR3 Q99500 4/20 0.39
S1PR4 O95977 1/20 0.37
S1PR5 Q9H228 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981614 0.89 S1PR1 (0.45) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1979486 0.87 S1PR1 (0.43) S1PR1S1PR3KDM4EMEN1CYP1A2
SCHEMBL12599365 0.84 NR1H2 (0.36) S1PR1MEN1KMT2A
SCHEMBL1981126 0.78 S1PR1 (0.50) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL2231440 0.76 S1PR1 (0.46) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1980001 0.76 S1PR1 (0.44) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL12522034 0.76 S1PR1 (0.53) S1PR1S1PR3S1PR4S1PR5
SCHEMBL1979890 0.76 S1PR1 (0.44) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL2230853 0.75 S1PR1 (0.49) S1PR1S1PR3S1PR4S1PR5KDM4E
SCHEMBL1979878 0.73 S1PR1 (0.49) S1PR1S1PR3S1PR4S1PR5KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP claimed
WO-2011069647-A1 NEW 2-AMINOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-06-16 WO claimed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed
WO-2011069647-A1 NEW 2-AMINOTHIADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-06-16 WO disclosed