SCHEMBL2230853

SCHEMBL2230853

CCCCN(Cc1ccccc1)c1nnc(-c2cc(C)c(OC)c(C)c2)s1.CCCCN(Cc1ccccc1F)c1nnc(-c2cc(C)c(OC)c(C)c2)s1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 11/20 0.49
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 1/20 0.43
UBE2N P61088 1/20 0.43
S1PR3 Q99500 5/20 0.40
LMNA P02545 1/20 0.37
S1PR4 O95977 1/20 0.36
S1PR5 Q9H228 1/20 0.36
CPB1 P15086 1/20 0.36
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
USP2 O75604 1/20 0.35
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981126 0.95 S1PR1 (0.50) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981536 0.92 S1PR1 (0.52) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1982705 0.85 S1PR1 (0.43) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981553 0.85 S1PR1 (0.51) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1981001 0.84 S1PR1 (0.46) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1980001 0.83 S1PR1 (0.44) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL2231440 0.83 S1PR1 (0.46) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1984811 0.82 S1PR1 (0.49) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1979878 0.82 S1PR1 (0.49) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10
SCHEMBL1980288 0.82 S1PR1 (0.41) S1PR1ALDH1A1KDM4ESMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP claimed
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed